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首页-小分子抑制剂&激动剂-Membrane Transporter/Ion Channel-GABA Transporter (GAT)-EF-1502
EF-1502

Chemical Structure : EF-1502

CAS No.: 684645-54-3

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EF-1502 (EF1502)

货号: PC-26893Not For Human Use, Lab Use Only.

EF-1502 (EF1502) is a selective inhibitor of GABA transporter GAT-1/BGT-1, noncompetitively inhibits both mGAT1 and the betaine/GABA transporter mGAT2 (BGT-1)) with Ki of 4 uM and 5 uM respectively, is inactive at GAT3 and GAT4.

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纯度 & COA & 质检文件 纯度: >98% (HPLC)

生物&药学活性

EF-1502 (EF1502) is a selective inhibitor of GABA transporter GAT-1/BGT-1, noncompetitively inhibits both mGAT1 and the betaine/GABA transporter mGAT2 (BGT-1)) with Ki of 4 uM and 5 uM respectively, is inactive at GAT3 and GAT4.

物理化学性质&存储条件

分子量 414.58
分子式 C22H26N2O2S2
外观性状 Solid
CAS No.
储存条件
固体粉末
-20°C 12 个月; 4°C 6 个月
配置液
-80°C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

4-((4,4-bis(3-methylthiophen-2-yl)but-3-en-1-yl)(methyl)amino)-4,5,6,7-tetrahydrobenzo[d]isoxazol-3-ol

参考文献

1. White HS, et al. J Pharmacol Exp Ther. 2005 Feb;312(2):866-74.

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