Darusentan | ETA receptor antagonist | Probechem Biochemicals

Chemical Structure : Darusentan

CAS No.: 171714-84-4

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Darusentan (Lu-135252, Lu 135252)

货号: PC-25045Not For Human Use, Lab Use Only.

Darusentan (Lu-135252) is a selective endothelin receptor A (ETA) receptor antagonist with binding Ki of 1.4 nM, >100-fold selective over ET-B receptor.

规格	价格	库存
5 mg	￥780	In stock
10 mg	￥1180	In stock
25 mg	￥1980	In stock
50 mg	￥3480	In stock
100 mg		Get quote

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生物&药学活性

Darusentan (Lu-135252) is a selective endothelin receptor A (ETA) receptor antagonist with binding Ki of 1.4 nM, >100-fold selective over ET-B receptor.

物理化学性质&存储条件

分子量	410.43
分子式	C22H22N2O6
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(S)-2-((4,6-Dimethoxypyrimidin-2-yl)oxy)-3-methoxy-3,3-diphenylpropanoic acid

参考文献

1. Frank Enseleit, et al. Ther Adv Cardiovasc Dis. 2010 Aug;4(4):231-40.

2. Liang F, et al. Can J Physiol Pharmacol. 2010 Aug;88(8):840-9.

Darusentan (Lu-135252, Lu 135252)

生物&药学活性

物理化学性质&存储条件

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Darusentan (Lu-135252, Lu 135252)

生物&药学活性

物理化学性质&存储条件

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