Darapladib |CAS:356057-34-6 Probechem Biochemicals

Chemical Structure : Darapladib

CAS No.: 356057-34-6

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货号: PC-42634Not For Human Use, Lab Use Only.

Darapladib (SB480848) is a potent Lp-PLA2 inhibitor with IC50 of 0.25 nM, shows an enhanced in vitro and in vivo profile versus SB-435495.

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Darapladib (SB480848) is a potent Lp-PLA2 inhibitor with IC50 of 0.25 nM, shows an enhanced in vitro and in vivo profile versus SB-435495.

分子量	666.7711
分子式	C36H38F4N4O2S
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	1H-Cyclopentapyrimidine-1-acetamide, N-[2-(diethylamino)ethyl]-2-[[(4-fluorophenyl)methyl]thio]-4,5,6,7-tetrahydro-4-oxo-N-[[4'-(trifluoromethyl)[1,1'-biphenyl]-4-yl]methyl]-

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3. Serruys PW, et al. Circulation. 2008 Sep 9;118(11):1172-82.