Dabigatran etexilate mesylate |CAS:872728-81-9 Probechem Biochemicals

Chemical Structure : Dabigatran etexilate mesylate

CAS No.: 872728-81-9

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Dabigatran etexilate mesylate (BIBR 1048MS;Dabigatran etexilate methanesulfonate)

货号: PC-42507Not For Human Use, Lab Use Only.

A prodrug of BIBR-953, which is a potent nonpeptide thrombin inhibitor with Ki of 4.5 nM.

规格	价格	库存
10 mg	￥560	In stock
50 mg	￥720	In stock
100 mg	￥960	In stock
200 mg		Get quote

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生物&药学活性

A prodrug of BIBR-953, which is a potent nonpeptide thrombin inhibitor with Ki of 4.5 nM; 10-fold less potent for Trypsin and no activity against Factor Xa, Plasmin, tPA and activated protein C; exhibits strong and long-lasting anticoagulant effects ex vivo and strong oral activity in different animal species.

Thrombosis

Approved

物理化学性质&存储条件

分子量	723.8389
分子式	C35H45N7O8S
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	β-Alanine, N-[[2-[[[4-[[[(hexyloxy)carbonyl]amino]iminomethyl]phenyl]amino]methyl]-1-methyl-1H-benzimidazol-5-yl]carbonyl]-N-2-pyridinyl-, ethyl ester, methanesulfonate (1:1)

参考文献

1. Hauel NH, et al. J Med Chem. 2002 Apr 25;45(9):1757-66.

2. Wienen W, et al. Thromb Haemost. 2007 Jul;98(1):155-62.

3. Baetz BE, et al. Pharmacotherapy. 2008 Nov;28(11):1354-73.

Dabigatran etexilate mesylate (BIBR 1048MS;Dabigatran etexilate methanesulfonate)

生物&药学活性

物理化学性质&存储条件

参考文献

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询单

Dabigatran etexilate mesylate (BIBR 1048MS;Dabigatran etexilate methanesulfonate)

生物&药学活性

物理化学性质&存储条件

参考文献

Bulk Inquiry

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询单

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