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首页-小分子抑制剂&激动剂-Epigenetics-Histone Acetyltransferase (HAT)-DS17701585
DS17701585

Chemical Structure : DS17701585

CAS No.: 2983027-66-1

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DS17701585 (DS 17701585)

货号: PC-38649Not For Human Use, Lab Use Only.

DS17701585 is a novel potent, highly selective EP300/CBP histone acetyltransferase inhibitor with IC50 of 0.15 uM.

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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

    生物&药学活性

    DS17701585 is a novel potent, highly selective EP300/CBP histone acetyltransferase inhibitor with IC50 of 0.15 uM.
    DS17701585 shows dose-dependent inhibition of SRY-box transcription factor 2 (SOX2) mRNA expression in a human lung squamous cell carcinoma cell line LK2-xenografted mouse model.

    物理化学性质&存储条件

    分子量 482.555
    分子式 C24H26N4O5S
    外观性状 Solid
    CAS No.
    储存条件
    固体粉末
    -20°C 12 个月; 4°C 6 个月
    配置液
    -80°C 6 个月; -20°C 6 个月
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    (S)-N-(1H-indazol-4-yl)-3-(1-(4-methoxyphenyl)cyclopentane-1-carbonyl)thiazolidine-4-carboxamide 1,1-dioxide

    参考文献

    1. Ryutaro Kanada, et al. Bioorg Med Chem Lett. 2022 Jun 15;66:128726.

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