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首页-小分子抑制剂&激动剂-Others-Other Targets-DS08701581
DS08701581

Chemical Structure : DS08701581

CAS No.:

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DS08701581 (DS 08701581)

货号: PC-22693Not For Human Use, Lab Use Only.

DS08701581 is a highly potent inhibitor of feline sarcoma-related (FER) tyrosine kinase with IC50 of 0.32 nM, shows in vivo antitumor efficacy.

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纯度 & COA & 质检文件 纯度: >98% (HPLC)

生物&药学活性

DS08701581 is a highly potent inhibitor of feline sarcoma-related (FER) tyrosine kinase with IC50 of 0.32 nM, shows in vivo antitumor efficacy.
DS08701581 shows potent cell-free and cell activities in this template, good oral BA, and improved kinase selectivity, resulting in significant tumor growth inhibition in the Ba/F3-FER tumor model without body weight loss.

物理化学性质&存储条件

分子量 488.60
分子式 C26H32N8O2
外观性状 Solid
CAS No.
储存条件
固体粉末
-20°C 12 个月; 4°C 6 个月
配置液
-80°C 6 个月; -20°C 6 个月
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Solubility

10 mM in DMSO
Chemical Name/SMILES

7-(((1R,2S)-2-aminocyclohexyl)amino)-5-((3-((2S,6R)-2,6-dimethylmorpholino)phenyl)amino)-4-oxo-3,4-dihydropyrido[3,4-d]pyridazine-8-carbonitrile

参考文献

1. Toru Taniguchi, et al. ACS Med Chem Lett. 2024 Jun 13;15(7):1010-1016.

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