DS-6930b | Probechem Biochemicals

Chemical Structure : DS-6930b

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DS-6930b (DS-6930 calcium salt;DS6930b)

货号: PC-35669Not For Human Use, Lab Use Only.

DS-6930b (DS-6930 calcium salt) is the calcium salt of DS-6930, which is a novel potent, selective PPARγ agonist with EC50 of 41 nM, Emax-68%.

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生物&药学活性

DS-6930b (DS-6930 calcium salt) is the calcium salt of DS-6930, which is a novel potent, selective PPARγ agonist with EC50 of 41 nM, Emax-68%.
DS-6930b significantly recruits several cofactors, such as RIP140 and PGC1, in cofactor recruitment assays.
DS-6930b demonstrates high PPARγ agonist potency with robust plasma glucose reduction, maintains diminished PPARγ-related adverse effects upon toxicological evaluation in vivo, and demonstrated no hepatotoxicity.

物理化学性质&存储条件

分子量
分子式
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	3-((6-((3,5-dimethylpyridin-2-yl)oxy)-1-methyl-1H-benzo[d]imidazol-2-yl)methoxy)benzoic acid 1/2 calcium

参考文献

1. Shinozuka T, et al. Bioorg Med Chem. 2018 Oct 1;26(18):5099-5117.

2. Shinozuka T, et al. Bioorg Med Chem. 2018 Oct 1;26(18):5079-5098.

DS-6930b (DS-6930 calcium salt;DS6930b)

生物&药学活性

物理化学性质&存储条件

参考文献

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DS-6930b (DS-6930 calcium salt;DS6930b)

生物&药学活性

物理化学性质&存储条件

参考文献

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