DS-6930 | PPARγ agonist | Probechem Biochemicals

Chemical Structure : DS-6930

加入收藏

DS-6930 (DS 6930;DS6930)

货号: PC-35674Not For Human Use, Lab Use Only.

DS-6930 (DS 6930, DS6930) is a novel potent, selective PPARγ agonist with EC50 of 41 nM, Emax-68%.

规格	价格	库存	数量
25 mg		Get quote
50 mg		Get quote
100 mg		Get quote

获取报价单

* 请选择数量再加入购物车

or Bulk Inquiry

大包装，大折扣！

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

生物&药学活性

DS-6930 (DS 6930, DS6930) is a novel potent, selective PPARγ agonist with EC50 of 41 nM, Emax-68%.
DS-6930 significantly recruits several cofactors, such as RIP140 and PGC1, in cofactor recruitment assays.
DS-6930 demonstrates high PPARγ agonist potency with robust plasma glucose reduction, maintains diminished PPARγ-related adverse effects upon toxicological evaluation in vivo, and demonstrated no hepatotoxicity.

物理化学性质&存储条件

分子量	403.438
分子式	C23H21N3O4
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	3-((6-((3,5-dimethylpyridin-2-yl)oxy)-1-methyl-1H-benzo[d]imidazol-2-yl)methoxy)benzoic acid calcium salt

参考文献

1. Shinozuka T, et al. Bioorg Med Chem. 2018 Oct 1;26(18):5099-5117.

2. Shinozuka T, et al. Bioorg Med Chem. 2018 Oct 1;26(18):5079-5098.

DS-6930 (DS 6930;DS6930)

生物&药学活性

物理化学性质&存储条件

参考文献

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

询单

DS-6930 (DS 6930;DS6930)

生物&药学活性

物理化学性质&存储条件

参考文献

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

询单

Get Quotation Now

* Indicates a Required FieldYour information is safe with us.