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首页-小分子抑制剂&激动剂-Epigenetics-Histone Methyltransferase (HMTase)-DC541
DC541

Chemical Structure : DC541

CAS No.: 2606862-00-2

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DC541 (DC 541)

货号: PC-38209Not For Human Use, Lab Use Only.

DC541 (DC 541) is a potent, selective peptidomimetic inhibitor of Protein N-terminal methyltransferase NTMT1 with IC50 of 0.34 uM.

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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

    生物&药学活性

    DC541 (DC 541) is a potent, selective peptidomimetic inhibitor of Protein N-terminal methyltransferase NTMT1 with IC50 of 0.34 uM.
    DC541 exhibits over 300-fold selectivity to several methyltransferases.
    DC541 inhibited funtions the cellular α-N-terminal methylation level of regulator of chromosome condensation 1 (RCC1, IC50 value of 30 μM) in human colorectal cancer HT29 cells.

    物理化学性质&存储条件

    分子量 529.641
    分子式 C30H35N5O4
    外观性状 Solid
    CAS No.
    储存条件
    固体粉末
    -20°C 12 个月; 4°C 6 个月
    配置液
    -80°C 6 个月; -20°C 6 个月
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    (S)-N-((S)-6-amino-1-((2-carbamoylphenyl)amino)-1-oxohexan-2-yl)-1-(2-(naphthalen-1-yl)acetyl)pyrrolidine-2-carboxamide

    参考文献

    1. Dongxing Chen, et al. ACS Med Chem Lett. 2021 Mar 1;12(3):485-493.

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