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首页-小分子抑制剂&激动剂-GPCR-Oxytocin Receptor (OXTR)-Cligosiban
Cligosiban

Chemical Structure : Cligosiban

CAS No.: 900510-03-4

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Cligosiban (PF-3274167;PF 03274167)

货号: PC-61369Not For Human Use, Lab Use Only.

Cligosiban (PF-3274167) is a potent, specific oxytocin receptor antagonist with Ki of 9.5 nM, displays high selectivity over the vasopressin receptors.

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10 mg ￥880 In stock
25 mg ￥1380 In stock
50 mg ￥2180 In stock
100 mg Get quote
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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

Cligosiban (PF-3274167) is a potent, specific oxytocin receptor antagonist with Ki of 9.5 nM, displays high selectivity over the vasopressin receptors.
Cligosiban (PF-3274167) demonstrates excellent potency and selectivity, as well as promising in vivo pharmacokinetics and significantly improved aqueous solubility.

物理化学性质&存储条件

分子量 419.841
分子式 C19H19ClFN5O3
外观性状 Solid
CAS No.
储存条件
固体粉末
-20 °C 12 个月; 4°C 6 个月
配置液
-80 °C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

5-(3-(3-(2-chloro-4-fluorophenoxy)azetidin-1-yl)-5-(methoxymethyl)-4H-1,2,4-triazol-4-yl)-2-methoxypyridine

参考文献

1. Vidal B, et al. Nucl Med Biol. 2017 Dec;55:1-6.

2. Brown A, et al. Bioorg Med Chem Lett. 2010 Jan 15;20(2):516-20.

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