Cilobradine |CAS:186097-54-1 Probechem Biochemicals

Chemical Structure : Cilobradine

CAS No.: 186097-54-1

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Cilobradine (DK-AH 269;DKAH-269)

货号: PC-45567Not For Human Use, Lab Use Only.

Cilobradine (DKAH-269) is a hyperpolarization-activated cyclic nucleotide-gated (HCN) channel, an open channel blocker of neuronal Ih and related cardiac If channels.

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生物&药学活性

Cilobradine (DKAH-269) is a hyperpolarization-activated cyclic nucleotide-gated (HCN) channel, an open channel blocker of neuronal Ih and related cardiac If channels.
Cilobradine (DKAH-269) strongly reduces the pacemaker diastolic depolarization rate and the cell's firing frequency.

物理化学性质&存储条件

分子量	519.0726
分子式	C28H39ClN2O5
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	100 mM in H2O (51.9 mg/mL)
Chemical Name/SMILES	2H-3-Benzazepin-2-one, 3-[[(3S)-1-[2-(3,4-dimethoxyphenyl)ethyl]-3-piperidinyl]methyl]-1,3,4,5-tetrahydro-7,8-dimethoxy-, hydrochloride (1:1)

参考文献

1. Van Bogaert PP, et al. Eur J Pharmacol. 2003 Oct 8;478(2-3):161-71.

2. El-Kholy W,et al. Mol Endocrinol. 2007 Mar;21(3):753-64.

3. Cheng Y, et al. J Pharmacol Exp Ther. 2007 May;321(2):469-76.

Cilobradine (DK-AH 269;DKAH-269)

生物&药学活性

物理化学性质&存储条件

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Cilobradine (DK-AH 269;DKAH-269)

生物&药学活性

物理化学性质&存储条件

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