欢迎访问ProbeChem中文网站，英文网站请访问www.probechem.com
    英文 |     中文

产品咨询: sales@probechem.com
订购: order@probechem.com

首页-小分子抑制剂&激动剂-Membrane Transporter/Ion Channel-GABA Receptor-Cenobamate
Cenobamate

Chemical Structure : Cenobamate

CAS No.: 913088-80-9

加入收藏

Cenobamate (YKP-3089, YKP3089)

货号: PC-28240Not For Human Use, Lab Use Only.

Cenobamate (YKP3089) is an antiepileptic compound that acts as a positive allosteric modulator of high-affinity GABAA receptors, potentiates GABA-induced currents (IGABA) in acutely isolated CA3 pyramidal cells with EC50 of 164 uM.

规格 价格 库存 数量
25 mg Get quote
50 mg Get quote
100 mg Get quote
获取报价单
* 请选择数量再加入购物车
 or Bulk Inquiry

大包装，大折扣！

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

纯度 & COA & 质检文件 纯度: >98% (HPLC)

生物&药学活性

Cenobamate (YKP3089) is an antiepileptic compound that acts as a positive allosteric modulator of high-affinity GABAA receptors, potentiates GABA-induced currents (IGABA) in acutely isolated CA3 pyramidal cells with EC50 of 164 uM.

物理化学性质&存储条件

分子量 267.67
分子式 C10H10ClN5O2
外观性状 Solid
CAS No.
储存条件
固体粉末
-20°C 12 个月; 4°C 6 个月
配置液
-80°C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

[(1R)-1-(2-chlorophenyl)-2-(tetrazol-2-yl)ethyl] carbamate

参考文献

1. Sperling MR, et al. Epilepsia. 2020 Jun;61(6):1099-1108.

2. Sharma R, et al. Eur J Pharmacol. 2020 Jul 15;879:173117.

3. Nakamura M, et al. Eur J Pharmacol. 2019 Jul 15;855:175-182.

备案号：沪ICP备16042516号-1 Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

联系我们 sales@probechem.com

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • *Additional Information:

询单

  • *产品名称:
  • *姓名:
  • *邮箱:
  • *公司名称:
  • *询单数量:
  • *国籍:
  • 询单信息: