Cangrelor | P2Y12 antagonist | Probechem Biochemicals

Chemical Structure : Cangrelor

CAS No.: 163706-06-7

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Cangrelor (AR-C69931MX)

货号: PC-61584Not For Human Use, Lab Use Only.

Cangrelor (AR-C69931MX) is a potent, selective P2T/P2Y12 receptor antagonist with IC50 of 0.4 nM against ADP-induced aggregation of human platelets.

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10 mg	￥1880	In stock
25 mg	￥2980	In stock
50 mg	￥4580	In stock
100 mg		Get quote

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生物&药学活性

Cangrelor (AR-C69931MX) is a potent, selective P2T/P2Y12 receptor antagonist with IC50 of 0.4 nM against ADP-induced aggregation of human platelets.
Cangrelor (AR-C69931MX) displays >1,000-fold selectivity over other P2 receptor family.
Cangrelor (AR-C69931MX) antagonizes the ex vivo and in vivo aggregatory actions of ADP, and displays a rapid onset and offset of action with the ability to prevent occlusive arterial thrombus formation.

物理化学性质&存储条件

分子量	776.36
分子式	C17H25Cl2F3N5O12P3S2
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	5'-Adenylic acid, N-[2-(methylthio)ethyl]-2-[(3,3,3-trifluoropropyl)thio]-, monoanhydride with (dichloromethylene)bis[phosphonic acid] (9CI)

参考文献

1. Ingall AH, et al. J Med Chem. 1999 Jan 28;42(2):213-20.

2. Huang J, et al. J Pharmacol Exp Ther. 2000 Nov;295(2):492-9.

3. Storey RF, et al. Br J Haematol. 2000 Sep;110(4):925-34.

Cangrelor (AR-C69931MX)

生物&药学活性

物理化学性质&存储条件

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Cangrelor (AR-C69931MX)

生物&药学活性

物理化学性质&存储条件

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