CYB210010 | 5-HT2 receptor agonist | Probechem Biochemicals

Chemical Structure : CYB210010

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CYB210010 (CYB-210010)

货号: PC-22124Not For Human Use, Lab Use Only.

CYB210010 is a potent and long-acting serotonin 5-HT2 receptor agonist with Ki values of 0.35 nM and 0.55 nM for 5-HT2A and 5-HT2C receptors respectively.

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生物&药学活性

CYB210010 is a potent and long-acting serotonin 5-HT2 receptor agonist with Ki values of 0.35 nM and 0.55 nM for 5-HT2A and 5-HT2C receptors respectively.
CYB210010 displays modest selectivity over 5-HT2B, 5-HT1A, 5-HT6, and adrenergic α2A receptors, and lacks activity at monoamine transporters and over 70 other proteins.
CYB210010 is orally bioavailable in three species, readily and preferentially crosses into the CNS, engages frontal cortex 5-HT2A receptors, and increases the expression of genes involved in neuroplasticity in the frontal cortex.
CYB210010 is a new tool molecule for investigating the therapeutic potential of 5-HT2 receptor activation.

物理化学性质&存储条件

分子量	281.29
分子式	C11H14F3NO2S
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	2-(2,5-dimethoxy-4-((trifluoromethyl)thio)phenyl)ethan-1-amine

参考文献

1. Geoffrey B Varty, et al. J Med Chem. 2024 Apr 9. doi: 10.1021/acs.jmedchem.3c01961.

CYB210010 (CYB-210010)

生物&药学活性

物理化学性质&存储条件

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CYB210010 (CYB-210010)

生物&药学活性

物理化学性质&存储条件

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