CVT-7124 | A2B adenosine receptor inhibitor | Probechem Biochemicals

Chemical Structure : CVT-7124

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CVT-7124 (CVT7124)

货号: PC-22012Not For Human Use, Lab Use Only.

CVT-7124 (CVT7124) is a highly potent, selective A2B adenosine receptor antagonist with Ki of 6 nM (hA2B), >830-fold selective over A1, A2A and A3 receptors.

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生物&药学活性

CVT-7124 (CVT7124) is a highly potent, selective A2B adenosine receptor antagonist with Ki of 6 nM (hA2B), >830-fold selective over A1, A2A and A3 receptors.
CVT-7124 blocks the release of interleukin-6 and monocyte chemotactic protein-1 from bronchial smooth muscle cells (BSMC).

物理化学性质&存储条件

分子量	404.35
分子式	C18H15F3N6O2
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	1-ethyl-8-(1-(3-(trifluoromethyl)benzyl)-1H-pyrazol-4-yl)-3,7-dihydro-1H-purine-2,6-dione

参考文献

1. Rao V Kalla, et al. Bioorg Med Chem Lett. 2008 Feb 15;18(4):1397-401.

CVT-7124 (CVT7124)

生物&药学活性

物理化学性质&存储条件

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CVT-7124 (CVT7124)

生物&药学活性

物理化学性质&存储条件

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