CV-6209 | PAF inhibitor | Probechem Biochemicals

Chemical Structure : CV-6209

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CV-6209 (CV 6209, CV6209)

货号: PC-60754Not For Human Use, Lab Use Only.

CV-6209 is a highly potent, selective platelet activating factor (PAF) inhibitor with IC50 of 75 and 170 nM for aggregation inhibition of rabbit and human platelets induced by PAF.

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生物&药学活性

CV-6209 is a highly potent, selective platelet activating factor (PAF) inhibitor with IC50 of 75 and 170 nM for aggregation inhibition of rabbit and human platelets induced by PAF.
CV-6209 shows little to no effects on the aggregation induced by arachidonic acid, ADP and collagen.
CV-6209 inhibited PAF-induced hypotension in rats (ED50=0.009 mg/kg i.v.) with no effect on the hypotension induced by arachidonic acid, histamine, bradykinin and isoproterenol.

物理化学性质&存储条件

分子量	642.3
分子式	C34H60N3O6Cl
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	2-[N-acetyl-N-(2-methoxy-3-octadecylcarbamoyloxypropoxycarbonyl) aminomethyl]-1-ethylpyridinium chloride

参考文献

1. Terashita Z, et al. J Pharmacol Exp Ther. 1987 Jul;242(1):263-8.

2. Terashita Z, et al. J Cardiovasc Pharmacol. 1988;12(5):505-11.

3. Stahl GL, et al. J Pharmacol Exp Ther. 1988 Mar;244(3):898-904.

4. Takatani M, et al. J Med Chem. 1989 Jan;32(1):56-64.

CV-6209 (CV 6209, CV6209)

生物&药学活性

物理化学性质&存储条件

参考文献

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CV-6209 (CV 6209, CV6209)

生物&药学活性

物理化学性质&存储条件

参考文献

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