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首页-小分子抑制剂&激动剂-GPCR-Opioid Receptor-CTAP TFA
CTAP TFA

Chemical Structure : CTAP TFA

CAS No.:

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CTAP TFA

货号: PC-27171Not For Human Use, Lab Use Only.

CTAP TFA is a potent, highly selective, and BBB-penetrant μ opioid receptor (MOR) antagonist with IC50 of 3.5 nM ,> 1200-fold selectivity over δ opioid receptor ( MOR, IC50=4500 nM) and somatostatin receptors.

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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

CTAP TFA is a potent, highly selective, and BBB-penetrant μ opioid receptor (MOR) antagonist with IC50 of 3.5 nM ,> 1200-fold selectivity over δ opioid receptor ( MOR, IC50=4500 nM) and somatostatin receptors.

物理化学性质&存储条件

分子量 1104.30 (free base)
分子式 C51H69N13O11S2.xC2HF3O2
外观性状 Solid
CAS No.
储存条件
固体粉末
-20°C 12 个月; 4°C 6 个月
配置液
-80°C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

{d-Phe}-Cys-Tyr-{d-Trp}-Arg-Thr-{Pen}-Thr-NH2 (Disulfide bridge:Cys2-Pen7) TFA salt

参考文献

1. Abbruscato TJ, et al. J Pharmacol Exp Ther. 1997 Jan;280(1):402-9.

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