CTA095 |CAS 1265823-05-9 Probechem Biochemicals

Chemical Structure : CTA095

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CTA095 (CTA 095;CTA-095)

货号: PC-35181Not For Human Use, Lab Use Only.

CTA095 (CTA-095) is a potent Etk (BMX) and Src dual inhibitor with IC50 of 60 and 120 nM, respectively, shows no significant inhibition on Btk and Yes at 10 uM.

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生物&药学活性

CTA095 (CTA-095) is a potent Etk (BMX) and Src dual inhibitor with IC50 of 60 and 120 nM, respectively, shows no significant inhibition on Btk and Yes at 10 uM.
CTA095 induces autophagy and apoptosis, as well as synergistic effects with autophagy modulators in prostate cancer cells.
CTA095 inhibits the phosphorylation of Etk, Src and the downstream signals Stat3 and Akt in prostate cancer cells.
CTA095nano inhibits PC3 xenograft tumor growth in vivo.

物理化学性质&存储条件

分子量	553.666
分子式	C35H31N5O2
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	2-(dibenzo[b,d]furan-2-yl)-7-phenyl-1-(3-(piperidin-1-yl)propyl)-1H-imidazo[4,5-g]quinoxalin-6(5H)-one

参考文献

1. Guo W, et al. PLoS One. 2013 Aug 15;8(8):e70910.

CTA095 (CTA 095;CTA-095)

生物&药学活性

物理化学性质&存储条件

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CTA095 (CTA 095;CTA-095)

生物&药学活性

物理化学性质&存储条件

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