CQ211 | RIOK2 inhibitor | Probechem Biochemicals

Chemical Structure : CQ211

CAS No.: 2648986-65-4

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CQ211 (CQ-211)

货号: PC-38737Not For Human Use, Lab Use Only.

CQ211 is a potent, highly selective RIOK2 (Right open reading frame kinase 2) inhibitor with Kd of 6.1 nM, shows excellent selectivity to RIOK2 in both enzymatic and cellular assays.

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10 mg	￥1280	In stock
25 mg	￥2180	In stock
50 mg	￥3580	In stock
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生物&药学活性

CQ211 is a potent, highly selective RIOK2 (Right open reading frame kinase 2) inhibitor with Kd of 6.1 nM, shows excellent selectivity to RIOK2 in both enzymatic and cellular assays.

CQ211 exhibits potent proliferation inhibition activity against multiple cancer cell lines (HT20, cell IC50=0.38 uM) and demonstrates promising in vivo efficacy in mouse xenograft models.

物理化学性质&存储条件

分子量	521.504
分子式	C26H22F3N7O2
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	8-(6-Methoxypyridin-3-yl)-1-(4-(piperazin-1-yl)-3-(trifluoromethyl)phenyl)-1,5-dihydro-4H-[1,2,3]triazolo[4,5-c]quinolin-4-on

参考文献

1. Yifan Ouyang, et al. J Med Chem. May 18, 2022.

CQ211 (CQ-211)

生物&药学活性

物理化学性质&存储条件

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CQ211 (CQ-211)

生物&药学活性

物理化学性质&存储条件

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