CPI-268456 |CAS:1380087-86-4 Probechem Biochemicals

Chemical Structure : CPI-268456

CAS No.: 1380087-86-4

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货号: PC-70026Not For Human Use, Lab Use Only.

CPI-268456 is a small molecule ligand of bromodomain-containing protein 4 (BRD4), binds to BRD4 with IC50 of 0.5 uM in cell-free assays.

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生物&药学活性

CPI-268456 is a small molecule ligand of bromodomain-containing protein 4 (BRD4), binds to BRD4 with IC50 of 0.5 uM in cell-free assays.

CPI-268456 inhibits LPS-induced IL-6 secretion in THP-1 cells with IC50 of 0.5 uM.

分子量	400.259
分子式	C20H15Cl2N3O2
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(S)-2-(8-chloro-6-(4-chlorophenyl)-1-methyl-4H-benzo[c]isoxazolo[4,5-e]azepin-4-yl)acetamide

1. Albrecht, B.K., Audia, J.E., Côté, A., et al. Bromodomain inhibitors and uses thereof. (2012).