CN750 |CAS:2098711-72-7 Probechem Biochemicals

Chemical Structure : CN750

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CN750 (CN-750;CN 750)

货号: PC-35750Not For Human Use, Lab Use Only.

CN750 (CN-750) is novel BRD4 (BD1, 2) inhibitor with IC50 of 44 nM, MV4-11 IC50 of 0.54 uM.

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生物&药学活性

CN750 (CN-750) is a potent BRD4 (BD1, 2) inhibitor with IC50 of 44 nM, MV4-11 IC50 of 0.54 uM.
CN750 shows Kd values of 33, 27, 24, 21, 20, 21, 18, 50, 20, 67, and 160 nM for BRD2 (BD1), BRD2 (BD1,2), BRD2 (BD2), BRD3 (BD1), BRD3 (BD1,2), BRD3 (BD2), BRD4 (BD1), BRD4 (BD2), BRDT (BD1), BRDT (BD1,2), and BRDT (BD2), respectively.
CN750 is a pan BET family inhibitor.

物理化学性质&存储条件

分子量	532.089
分子式	C29H34ClN7O
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	5-(4-((3-chlorobenzyl)amino)-2-(4-(2-(dimethylamino)ethyl)piperazin-1-yl)quinazolin-6-yl)-1-methylpyridin-2(1H)-one

参考文献

1. Yang SM, et al. Bioorg Med Chem Lett. 2018 Nov 15;28(21):3483-3488.

CN750 (CN-750;CN 750)

生物&药学活性

物理化学性质&存储条件

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CN750 (CN-750;CN 750)

生物&药学活性

物理化学性质&存储条件

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