欢迎访问ProbeChem中文网站，英文网站请访问www.probechem.com
    英文 |     中文

产品咨询: sales@probechem.com
订购: order@probechem.com

首页-小分子抑制剂&激动剂-Apoptosis-DAPK-CK156
CK156

Chemical Structure : CK156

CAS No.: 2910938-59-7

加入收藏

CK156 (CK-156)

货号: PC-38745Not For Human Use, Lab Use Only.

CK156 is a potent, highly selective serine/threonine kinase 17A (DRAK1) inhibitor with Kd of 21 nM, cellular IC50 of 182 nM.

规格 价格 库存 数量
10 mg Get quote
25 mg Get quote
50 mg Get quote
获取报价单
* 请选择数量再加入购物车
 or Bulk Inquiry

大包装，大折扣！

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

    生物&药学活性

    CK156 is a potent, highly selective serine/threonine kinase 17A (STK17A, DRAK1) inhibitor with Kd of 21 nM, cellular IC50 of 182 nM.
    CK156 demonstrates excellent selectivity in kinomewide screens.
    CK156 inhibits cell growth of glioma cells in 2D and 3D culture only at low micromolar concentrations.

    物理化学性质&存储条件

    分子量 395.463
    分子式 C21H25N5O3
    外观性状 Solid
    CAS No.
    储存条件
    固体粉末
    -20°C 12 个月; 4°C 6 个月
    配置液
    -80°C 6 个月; -20°C 6 个月
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    (13Z,14E)-N-(tert-butyl)-3,6-dioxa-9-aza-1(3,5)-pyrazolo[1,5-a]pyrimidina-2(1,3)-benzenacyclononaphane-24-carboxamide

    参考文献

    1. Christian G Kurz, et al. J Med Chem. 2022 May 24. doi: 10.1021/acs.jmedchem.2c00173.

    备案号：沪ICP备16042516号-1 Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

    联系我们 sales@probechem.com

    Bulk Inquiry

    * Indicates a Required FieldYour information is safe with us.

    • *Product name:
    • *Applicant name:
    • *Email address:
    • *Organization name:
    • *Requested quantity:
    • *Country:
    • *Additional Information:

    询单

    • *产品名称:
    • *姓名:
    • *邮箱:
    • *公司名称:
    • *询单数量:
    • *国籍:
    • 询单信息: