CCG 258748 |CAS: 2410997-49-6 Probechem Biochemicals

Chemical Structure : CCG 258748

加入收藏

CCG 258748 (CCG258748;CCG-258748)

货号: PC-60586Not For Human Use, Lab Use Only.

CCG 258748 is a potent, selective G protein-coupled receptor kinase GRK2 inhibitor with IC50 of 8 nM.

规格	价格	库存	数量
50 mg		Get quote
100 mg		Get quote
250 mg		Get quote

获取报价单

* 请选择数量再加入购物车

or Bulk Inquiry

大包装，大折扣！

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

生物&药学活性

CCG 258748 is a potent, selective G protein-coupled receptor kinase GRK2 inhibitor with IC50 of 8 nM.
CCG 258748 displays 30-fold selectivity over GRK5, and no significant inhibitory activity against GRK1, PKA and ROCK1.

物理化学性质&存储条件

分子量	448.502
分子式	C24H25FN6O2
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	5-((3S,4R)-3-(((1H-indazol-5-yl)oxy)methyl)piperidin-4-yl)-N-((1H-pyrazol-5-yl)methyl)-2-fluorobenzamide

参考文献

1. Bouley R, et al. Mol Pharmacol. 2017 Dec;92(6):707-717.

CCG 258748 (CCG258748;CCG-258748)

生物&药学活性

物理化学性质&存储条件

参考文献

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

询单

CCG 258748 (CCG258748;CCG-258748)

生物&药学活性

物理化学性质&存储条件

参考文献

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

询单

Get Quotation Now

* Indicates a Required FieldYour information is safe with us.