CCG258208 hydrochloride

Chemical Structure : CCG258208 hydrochloride

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货号: PC-23975Not For Human Use, Lab Use Only.

CCG258208 hydrochloride is a potent selective GRK2 inhibitor with IC50 of 30 nM, >200-fold selectivity over GRK1 and GRK5.

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CCG258208 hydrochloride is a potent selective GRK2 inhibitor with IC50 of 30 nM, >200-fold selectivity over GRK1 and GRK5.

分子量	488.94
分子式	C24H26ClFN4O4
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
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Solubility	10 mM in DMSO
Chemical Name/SMILES	Benzamide, 5-[(3S,4R)-3-[(1,3-benzodioxol-5-yloxy)methyl]-4-piperidinyl]-2-fluoro-N-(1H-pyrazol-3-ylmethyl)- hydrochloride

1. Bouley RA, et al. Mol Pharmacol. 2020 Jun;97(6):392-401.