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首页-小分子抑制剂&激动剂-Others-GRK (GPCRK)-CCG215022
CCG215022

Chemical Structure : CCG215022

CAS No.: 1813527-81-9

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CCG215022 (CCG-215022, CCG 215022)

货号: PC-45591Not For Human Use, Lab Use Only.

CCG-215022 (CCG215022) is a potent and selective pan GRK (G protein-coupled receptor kinase) inhibitor with IC50 of 0.15/0.38/3.9 uM for GRK2/5/1 respectively.

规格 价格 库存 数量
2 mg ￥1280 In stock
5 mg ￥2180 In stock
10 mg ￥3580 In stock
50 mg Get quote
100 mg Get quote
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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

CCG215022 (CCG-215022) is a potent and selective pan GRK (G protein-coupled receptor kinase) inhibitor with IC50 of 0.15/0.38/3.9 uM for GRK2/5/1 respectively.
CCG215022 displays 300-800 fold selectivity against PKA.
CCG215022 exhibits improved potency compared with GSK180736A.

物理化学性质&存储条件

分子量 499.4964
分子式 C26H22FN7O3
外观性状 Solid
CAS No.
储存条件
固体粉末
-20 °C 12 个月; 4°C 6 个月
配置液
-80 °C 6 个月; -20°C 6 个月
Shipping
Solubility

DMSO: ≥ 28 mg/mL
Chemical Name/SMILES

4-(4-fluoro-3-((pyridin-2-ylmethyl)carbamoyl)phenyl)-N-(1H-indazol-5-yl)-6-methyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide

参考文献

1. Homan KT, et al. J Biol Chem. 2015 Aug 21;290(34):20649-59.

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