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首页-小分子抑制剂&激动剂-Others-Regulators of G protein signaling (RGS)-CCG-63808
CCG-63808

Chemical Structure : CCG-63808

CAS No.: 620113-73-7

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CCG-63808 (CCG63808, CCG 63808)

货号: PC-45956Not For Human Use, Lab Use Only.

A reversible, allosteric inhibitor of regulator of G-protein signaling (RGS) proteins with a potency order of RGS4 >19=16>8>>7.

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5 mg ￥880 In stock
10 mg ￥1380 In stock
25 mg ￥2580 In stock
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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

CCG-63808 is a reversible, allosteric inhibitor of regulator of G-protein signaling (RGS) proteins with a potency order of RGS4 >19=16>8>>7.
CCG-63808 inhibits the Gαo-RGS4 interaction with IC50 of 1.9 uM, does not inhibit Gα binding to RGS7, 2- to 10-fold more potent at RGS4 than on the other closely related R4 family members, RGS8 and RGS16.

物理化学性质&存储条件

分子量 454.4756
分子式 C25H15FN4O2S
外观性状 Solid
CAS No.
储存条件
固体粉末
-20 °C 12 个月; 4°C 6 个月
配置液
-80 °C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

2-Benzothiazoleacetonitrile, .alpha.-[[2-(4-fluorophenoxy)-9-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-3-yl]methylene]-

参考文献

1. Blazer LL, et al. Mol Pharmacol. 2010 Sep;78(3):524-33.

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