CAMKK2 inhibitor 4t |CAS: 2230039-14-0 Probechem Biochemicals

Chemical Structure : CAMKK2 inhibitor 4t

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CAMKK2 inhibitor 4t

货号: PC-63352Not For Human Use, Lab Use Only.

CAMKK2 inhibitor 4t is a potent, selective, orally available, brain-penetrant CAMKK2 inhibitor with pIC50 of 8.5.

规格	价格	库存	数量
25 mg		Get quote
100 mg		Get quote
250 mg		Get quote
1 g		Get quote

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生物&药学活性

CAMKK2 inhibitor 4t is a potent, selective, orally available, brain-penetrant CAMKK2 inhibitor with pIC50 of 8.5.
CAMKK2 inhibitor 4t potently inhibits AMPK phosphorylation in a hypothalamus-derived cell line with pIC50 of 6.3; reduces food intake in rodent models.

物理化学性质&存储条件

分子量	480.612
分子式	C30H32N4O2
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	2-isopropyl-4-(2-(2-methyl-4-(2-morpholinoethoxy)phenyl)-1H-pyrrolo[2,3-b]pyridin-4-yl)benzonitrile

参考文献

1. Price DJ, et al. Bioorg Med Chem Lett. 2018 Apr 5. pii: S0960-894X(18)30223-3.