Bromocriptine mesylate |CAS:22260-51-1 Probechem Biochemicals

Chemical Structure : Bromocriptine mesylate

CAS No.: 22260-51-1

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Bromocriptine mesylate (CB-154)

货号: PC-43160Not For Human Use, Lab Use Only.

Bromocriptine (CB-154) is a dopamine D2 receptor agonist (Ki=3 nM) and and various serotonin receptors, also inhibits the release of glutamate by reversing the glutamate GLT1 transporter.

规格	价格	库存
100 mg	￥680	In stock
250 mg	￥1180	In stock
500 mg	￥1980	In stock
1 g		Get quote

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生物&药学活性

Bromocriptine (CB-154) is a dopamine D2 receptor agonist (Ki=3 nM) and and various serotonin receptors, also inhibits the release of glutamate by reversing the glutamate GLT1 transporter.
Bromocriptine (CB-154) decreases body fat in animal and human models and increases lean muscle mass, improves glucose intolerance and insulin resistance, and reduces triglycerides and free fatty acids.
Bromocriptine (CB-154) also induces apoptosis and decreases colony formation in AML cells, shows synergy with standard agents and selectivity for the leukemic cell.
Bromocriptine (CB-154) reduces hyperphagia and adiposity in rats with diet-induced obesity.

物理化学性质&存储条件

分子量	750.7001
分子式	C33H44BrN5O8S
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	DMSO: ≥ 30 mg/mL
Chemical Name/SMILES	Ergotaman-3',6',18-trione, 2-bromo-12'-hydroxy-2'-(1-methylethyl)-5'-(2-methylpropyl)-, (5α)-, methanesulfonate (1:1)

参考文献

1. Shirasaki Y, et al. Eur J Pharmacol. 2010 Sep 15;643(1):48-57.

2. Oda T, et al. Eur J Pharmacol. 2008 Nov 19;598(1-3):27-31.

3. Wacker J, et al. Psychophysiology. 2006 Jul;43(4):372-81.

4. Liberante FG, et al. Oncotarget. 2016 Feb 9;7(6):6609-19.

Bromocriptine mesylate (CB-154)

生物&药学活性

物理化学性质&存储条件

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Bromocriptine mesylate (CB-154)

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物理化学性质&存储条件

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