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首页-小分子抑制剂&激动剂-Epigenetics-Histone Demethylase-Bizine
Bizine

Chemical Structure : Bizine

CAS No.: 1591932-50-1

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Bizine

货号: PC-62871Not For Human Use, Lab Use Only.

Bizine is a phenelzine analog that inhibits LSD1 with Ki of 59 nM, displays 23-fold, 63-fold, and >100-fold selectivity for LSD-1 over MAOA, MAOB, and LSD2 respectively.

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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

    生物&药学活性

    Bizine is a phenelzine analog that inhibits LSD1 with Ki of 59 nM, displays 23-fold, 63-fold, and >100-fold selectivity for LSD-1 over MAOA, MAOB, and LSD2 respectively.
    Bizine induces bulk histone H3 lysine 4 dimethylation in LNCaP cancer cells (EC50=2 uM).
    Bizine protects neurons exposed to oxidative stress at 0.5 uM.

    物理化学性质&存储条件

    分子量 297.402
    分子式 C18H23N3O
    外观性状 Solid
    CAS No.
    储存条件
    固体粉末
    -20 °C 12 个月; 4°C 6 个月
    配置液
    -80 °C 6 个月; -20°C 6 个月
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    N-[4-(2-hydrazinylethyl)phenyl]-benzenebutanamide

    参考文献

    1. Prusevich P, et al. ACS Chem Biol. 2014 Jun 20;9(6):1284-93.

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