Bivalirudin | Thrombin inhibitor | Probechem Biochemicals

Chemical Structure : Bivalirudin

CAS No.: 128270-60-0

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Bivalirudin (Bivalitroban)

货号: PC-73174Not For Human Use, Lab Use Only.

Bivalirudin (Bivalitroban) is a potent, selective inhibitor of α- and ζ-thrombin (Ki= 2.56 and 1.84 nM, respectively), exhibits high fibrinogen-clotting activities.

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25 mg	￥1580	In stock
100 mg	￥3580	In stock
500 mg	￥7580	In stock
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生物&药学活性

Bivalirudin (Bivalitroban) is a potent, selective inhibitor of α- and ζ-thrombin (Ki= 2.56 and 1.84 nM, respectively), exhibits high fibrinogen-clotting activities.
Bivalirudin displays >1,000-fold selecivity for α- and ζ-thrombin over trypsin and γ-thrombin.
Bivalirudin inhibits α-thrombin-stimulated activation of the clotting factors Factor X, Factor V, and prothrombin in contact-activated plasma at 0.1 uM.
Bivalirudin (0.5-1.5 mg/kg, i.v.) reduces platelet deposition in a rat carotid endarterectomy model in a dose-dependent manner.

物理化学性质&存储条件

分子量	2180.3
分子式	C98H138N24O33
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 Month
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Solubility
Chemical Name/SMILES

参考文献

1. Witting, J.I., et al. Biochem J. 283(Pt 3), 737-743 (1992).

2. Ofosu, F.A., et al. Biochem J. 283(Pt 3), 893-897 (1992).

3. Hamelink, J.K., et al. J. Vasc. Surg. 21(3), 492-498 (1995).

Bivalirudin (Bivalitroban)

生物&药学活性

物理化学性质&存储条件

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Bivalirudin (Bivalitroban)

生物&药学活性

物理化学性质&存储条件

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