BRPF1B TRIM24-IN-34 |CAS:1242907-48-7 Probechem Biochemicals

Chemical Structure : BRPF1B TRIM24-IN-34

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BRPF1B TRIM24-IN-34

货号: PC-62285Not For Human Use, Lab Use Only.

BRPF1B TRIM24-IN-34 is a selective BRPF1B/TRIM24 dual inhibitor that binds with KD of 137 and 222 nM, respectively.

规格	价格	库存	数量
25 mg		Get quote
100 mg		Get quote
200 mg		Get quote
1 g		Get quote

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生物&药学活性

BRPF1B TRIM24-IN-34 is a selective BRPF1B/TRIM24 dual inhibitor that binds with KD of 137 and 222 nM, respectively.
BRPF1B TRIM24-IN-34 exhibits good selectivity over other bromodomains.
BRPF1B TRIM24-IN-34 showes no significant cytotoxicity in a panel of cancer cell lines (GI50>10 uM).

物理化学性质&存储条件

分子量	499.538
分子式	C24H25N3O7S
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	3,4-dimethoxy-N-(6-(4-methoxyphenoxy)-1,3-dimethyl-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-5-yl)benzenesulfonamide

参考文献

1. Bennett J, et al. J Med Chem. 2016 Feb 25;59(4):1642-7.