BRD9-IN-28 |CAS:1947372-67-9 Probechem Biochemicals

Chemical Structure : BRD9-IN-28

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BRD9-IN-28

货号: PC-62938Not For Human Use, Lab Use Only.

BRD9-IN-28 is a highly potent and selective BRD7/9 bromodomain inhibitor with pIC50 of 6.9, Kd of 68 nM for BRD9.

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生物&药学活性

BRD9-IN-28 is a highly potent and selective BRD7/9 bromodomain inhibitor with pIC50 of 6.9, Kd of 68 nM for BRD9.
BRD9-IN-28 is slightly less potent against BRD7 (Kd=368 nM) and completely inactive against BAZ2B, little affinity across BRD proteins from sub-families 1-3 and 5-8, including BAZ2A and BAZ2B.
BRD9-IN-28 shows weak affinity for the BRDs from CBP, p300 and FALZ.

物理化学性质&存储条件

分子量	360.417
分子式	C21H20N4O2
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	1-(1-(imidazo[1,2-a]pyridin-5-yl)-7-morpholinoindolizin-3-yl)ethan-1-one

参考文献

1. Duncan. A. Hay, et al. Med. Chem. Commun., 2015, DOI: 10.1039/C5MD00152H.

BRD9-IN-28

生物&药学活性

物理化学性质&存储条件

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BRD9-IN-28

生物&药学活性

物理化学性质&存储条件

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