BMS-986122 |CAS:313669-88-4 Probechem Biochemicals

Chemical Structure : BMS-986122

CAS No.: 313669-88-4

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BMS-986122 (BMS986122)

货号: PC-63080Not For Human Use, Lab Use Only.

BMS-986122 is a potent positive allosteric modulator of μ-opioid (MOR) receptor, significantly increases the inhibition of forskolin-stimulated adenylyl cyclase activity produced by an EC10 (30 pM) concentration of endomorphin-I in CHO-μ cells.

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5 mg	￥1280	In stock
10 mg	￥1980	In stock
25 mg	￥3280	In stock
50 mg		Get quote
100 mg		Get quote

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生物&药学活性

BMS-986122 is a potent positive allosteric modulator of μ-opioid (MOR) receptor, significantly increases the inhibition of forskolin-stimulated adenylyl cyclase activity produced by an EC10 (30 pM) concentration of endomorphin-I in CHO-μ cells.

物理化学性质&存储条件

分子量	448.774
分子式	C16H15BrClNO3S2
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	2-(3-Bromo-4-methoxyphenyl)-3-[(4-chlorophenyl)sulfonyl]-thiazolidine

参考文献

1. Burford NT, et al. Proc Natl Acad Sci U S A. 2013 Jun 25;110(26):10830-5.

2. Livingston KE, et al. Proc Natl Acad Sci U S A. 2014 Dec 23;111(51):18369-74.

3. Livingston KE, et al. Mol Pharmacol. 2018 Feb;93(2):157-167.

BMS-986122 (BMS986122)

生物&药学活性

物理化学性质&存储条件

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BMS-986122 (BMS986122)

生物&药学活性

物理化学性质&存储条件

参考文献

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