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首页-小分子抑制剂&激动剂-GPCR-Melanin-concentrating Hormone Receptor (MCHR)-BMS-819881
BMS-819881

Chemical Structure : BMS-819881

CAS No.: 1197420-05-5

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BMS-819881 (BMS819881)

货号: PC-61121Not For Human Use, Lab Use Only.

A potent, selective melanin concentrating hormone receptor 1 (MCHR1) inhibitor with Ki of 10.4 nM.

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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

    生物&药学活性

    BMS-819881 is a potent, selective melanin concentrating hormone receptor 1 (MCHR1) inhibitor with Ki of 10.4 nM.
    BMS-819881 effectively blocks MCH stimulated Ca+2 mobilization in heterologous cells overexpressing MCHR1 but not the cells expressing MCHR2 at 10 uM.
    BMS-819881 shows potential for treatment of obesity.

    物理化学性质&存储条件

    分子量 468.952
    分子式 C24H21ClN2O4S
    外观性状 Solid
    CAS No.
    储存条件
    固体粉末
    -20 °C 12 个月; 4°C 6 个月
    配置液
    -80 °C 6 个月; -20°C 6 个月
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    (R)-6-(4-chlorophenyl)-3-(4-(2-cyclopropyl-2-hydroxyethoxy)-3-methoxyphenyl)-thieno[3,2-d]pyrimidin-4(3H)-one

    参考文献

    1. Washburn WN, et al. J Med Chem. 2014 Sep 25;57(18):7509-22.

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