BMS-795311 |CAS:939390-99-5 Probechem Biochemicals

Chemical Structure : BMS-795311

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BMS-795311 (BMS795311)

货号: PC-63563Not For Human Use, Lab Use Only.

BMS-795311 is a potent and orally available CETP inhibitor with IC50 of 3.8 nM, inhibits cholesteryl ester (CE) transfer with IC50 of 0.22 uM.

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生物&药学活性

BMS-795311 is a potent and orally available CETP inhibitor with IC50 of 3.8 nM, inhibits cholesteryl ester (CE) transfer with IC50 of 0.22 uM.
BMS-795311 inhibits CE transfer activity at an oral dose of 1 mg/kg in human CETP/apoB-100 dual transgenic mice and increased HDL cholesterol content and size comparable to Torcetrapib in moderately-fat fed hamsters.

物理化学性质&存储条件

分子量	671.535
分子式	C33H23F10NO3
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
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Solubility	10 mM in DMSO
Chemical Name/SMILES	N-[(1R)-1-(3-Cyclopropoxy-4-fluorophenyl)-1-[3-fluoro-5-(1,1,2,2-tetrafluoroethoxy)phenyl]-2-phenylethyl]-4-fluoro-3-(trifluoromethyl)benzamide

参考文献

1. Qiao JX, et al. J Med Chem. 2015 Nov 25;58(22):9010-26.

BMS-795311 (BMS795311)

生物&药学活性

物理化学性质&存储条件

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BMS-795311 (BMS795311)

生物&药学活性

物理化学性质&存储条件

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