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首页-小分子抑制剂&激动剂-GPCR-Melanocortin Receptor-BL-6020 979
BL-6020 979

Chemical Structure : BL-6020 979

CAS No.:

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BL-6020 979 (SNT207979;BL-6020/979)

货号: PC-61572Not For Human Use, Lab Use Only.

BL-6020/979 (SNT207979) is an orally available, selective, potent MC4R antagonist with IC50 of 19 nM.

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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

    生物&药学活性

    BL-6020/979 (SNT207979) is an orally available, selective, potent MC4R antagonist with IC50 of 19 nM.
    BL-6020/979 (SNT207979) weakly binds to MC-3 and MC-5 receptors with IC50 of 2.7 uM and 0.89 uM, respectively, >10,000-fold selectivity over MC-1R;.
    BL-6020/979 (SNT207979) demonstrates in animal models and presents a promising candidate suitable for further development towards a first-in-class treatment option for cachexia.

    物理化学性质&存储条件

    分子量
    分子式
    外观性状 Solid
    CAS No.
    储存条件
    固体粉末
    -20 °C 12 个月; 4°C 6 个月
    配置液
    -80 °C 6 个月; -20°C 6 个月
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    参考文献

    1. Dallmann R, et al. J Cachexia Sarcopenia Muscle. 2011 Sep;2(3):163-174.

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