BI 6901 |CAS:2040401-92-9 Probechem Biochemicals

Chemical Structure : BI 6901

CAS No.: 2040401-92-9

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BI 6901 (BI6901)

货号: PC-35030Not For Human Use, Lab Use Only.

BI 6901 is a potent, selective CCR10 antagonist with Aequorin Ca2+ flux pIC50 of 9.0, shows high selectivity over other GPCRs.

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5 mg	￥3580	In stock
10 mg	￥5580	In stock
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生物&药学活性

BI 6901 is a potent, selective CCR10 antagonist with Aequorin Ca2+ flux pIC50 of 9.0, shows high selectivity over other GPCRs.
BI 6901 inhibits the CCL27 dependent chemotaxis of Ba/F3 cells stably transfected with human CCR10 with pIC50 of 9.0.
BI 6901 is efficacious in a murine model of DNFB contact hypersensitivity, inhibits DNFB stimulated inflammatory response in sensitized Balb-C mice.

物理化学性质&存储条件

分子量	453.561
分子式	C23H27N5O3S
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	N-[(2R)-4-(2-cyanopyrrol-1-yl)-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl]-1H-indole-4-sulfonamide

参考文献

1. Abeywardane A, et al. Bioorg Med Chem Lett. 2016 Nov 1;26(21):5277-5283.

BI 6901 (BI6901)

生物&药学活性

物理化学性质&存储条件

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BI 6901 (BI6901)

生物&药学活性

物理化学性质&存储条件

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