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首页-小分子抑制剂&激动剂-Membrane Transporter/Ion Channel-TRP Channel-BCTC
BCTC

Chemical Structure : BCTC

CAS No.: 393514-24-4

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BCTC (TRPV1 antagonist)

货号: PC-45764Not For Human Use, Lab Use Only.

BCTC is a highly potent, selective, CNS-penetrant TRPV1 antagonist that inhibits capsaicin-induced and acid-induced activation of rat TRPV1 with IC50 values of 35 and 6 nM, respectively.

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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

BCTC is a highly potent, selective, CNS-penetrant TRPV1 antagonist that inhibits capsaicin-induced and acid-induced activation of rat TRPV1 with IC50 values of 35 and 6 nM, respectively.
BCTC shows selectivity against 63 other receptor, enzyme, transporter, and ion channel targets; orally bioavailable.

物理化学性质&存储条件

分子量 372.8917
分子式 C20H25ClN4O
外观性状 Solid
CAS No.
储存条件
固体粉末
-20 °C 12 个月; 4°C 6 个月
配置液
-80 °C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

1-Piperazinecarboxamide, 4-(3-chloro-2-pyridinyl)-N-[4-(1,1-dimethylethyl)phenyl]-

参考文献

1. Valenzano KJ, et al. J Pharmacol Exp Ther. 2003 Jul;306(1):377-86.

2. Gavva NR, et al. Mol Pharmacol. 2005 Dec;68(6):1524-33.

3. Yamamoto M, et al. World J Gastroenterol. 2016 Nov 28;22(44):9752-9764.

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