TP-021 (BCL6 inhibitor 8c) |CAS:2130878-25-8 Probechem Biochemicals

Chemical Structure : BCL6 inhibitor 8c

CAS No.: 2130878-25-8

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BCL6 inhibitor 8c (TP-021, BCL6-IN-8c)

货号: PC-61016Not For Human Use, Lab Use Only.

TP-021 (BCL6 inhibitor 8c) is a potent, in vivo-active BCL6 inhibitor with IC50 of 0.1 uM in ELISA assays.

规格	价格	库存
5 mg	￥1980	In stock
10 mg	￥2980	In stock
25 mg	￥4980	In stock
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100 mg		Get quote

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生物&药学活性

TP-021 (BCL6 inhibitor 8c) is a potent, in vivo-active BCL6 inhibitor with IC50 of 0.1 uM in ELISA assays.
BCL6 inhibitor 8c exhibits good cellular BCL6BTB/ BCoR PPI inhibitory activity in the submicromolar range (M2H IC50=0.72 uM).
BCL6 inhibitor 8c showed a good pharmacokinetic profile, which is acceptable for both in vitro and in vivo studies.

物理化学性质&存储条件

分子量	417.846
分子式	C20H20ClN3O5
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
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Solubility	10 mM in DMSO
Chemical Name/SMILES	6-((2-Chloro-4-nitro-5-((tetrahydro-2H-pyran-4-yl)oxy)phenyl)amino)-3,4-dihydroquinolin-2(1H)-one

参考文献

1. Yasui T, et al. Bioorg Med Chem. 2017 Sep 1;25(17):4876-4886.

BCL6 inhibitor 8c (TP-021, BCL6-IN-8c)

生物&药学活性

物理化学性质&存储条件

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BCL6 inhibitor 8c (TP-021, BCL6-IN-8c)

生物&药学活性

物理化学性质&存储条件

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