BCAT2-IN-1 | BACT2 inhibitor | Probechem Biochemicals

Chemical Structure : BCAT2-IN-1

CAS No.: 1875078-61-7

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BCAT2-IN-1 (BCATm inhibitor)

货号: PC-26618Not For Human Use, Lab Use Only.

BCAT2-IN-1 is a potent, selective, in-vivo efficacious BCATm (BCAT2) inhibitor with pIC50 of 7.3, 100-fold selective for BCATm over BCATc.

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5 mg	￥1780	In stock
10 mg	￥2780	In stock
25 mg	￥4980	In stock
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100 mg		Get quote

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生物&药学活性

BCAT2-IN-1 is a potent, selective, in-vivo efficacious BCATm (BCAT2) inhibitor with pIC50 of 7.3, 100-fold selective for BCATm over BCATc.
BCAT2-IN-1 binds to the active site of BACTm in a unique mode via multiple H-bond and van der Waals interactions.
BCAT2-IN-1 effectively raised the levels of BCAAs in an acute animal model over an extended duration.

物理化学性质&存储条件

分子量	538.46
分子式	C25H24BrN5O2S
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	1H-Benzimidazole-5-carboxamide, 1-[(1R,3S)-3-[[(5-bromo-2-thienyl)carbonyl]amino]cyclohexyl]-N-methyl-2-(2-pyridinyl)-, rel-

参考文献

1. Hongfeng Deng, et al. ACS Med Chem Lett. 2016 Feb 8;7(4):379-84.

BCAT2-IN-1 (BCATm inhibitor)

生物&药学活性

物理化学性质&存储条件

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BCAT2-IN-1 (BCATm inhibitor)

生物&药学活性

物理化学性质&存储条件

参考文献

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