BAY-6035 |CAS: 2247890-13-5 Probechem Biochemicals

Chemical Structure : BAY-6035

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BAY-6035 (BAY6035)

货号: PC-63250Not For Human Use, Lab Use Only.

BAY-6035 is a potent, peptide-competitive inhibitor of histone methyltransferase SMYD3, inhibits in vitro methylation of MEKK2 peptide with IC50 of 88 nM, >100-fold selectivity over other HMTases.

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生物&药学活性

BAY-6035 is a potent, peptide-competitive inhibitor of histone methyltransferase SMYD3, inhibits in vitro methylation of MEKK2 peptide with IC50 of 88 nM, >100-fold selectivity over other HMTases; inhibits the methylation of MEKK2 in cells with IC50 of 70 nM.

物理化学性质&存储条件

分子量	396.491
分子式	C22H28N4O3
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(2S)-1-(3-azabicyclo[3.1.0]hexane-3-carbonyl)-N-(2-cyclopropylethyl)-2-methyl-4-oxo-2,3,4,5-tetrahydro-1H-benzo[b][1,4]diazepine-7-carboxamide

参考文献

1, Stefan Gradl, et al. SLAS Discov. 2021 Sep;26(8):947-960.

BAY-6035 (BAY6035)

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物理化学性质&存储条件

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BAY-6035 (BAY6035)

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物理化学性质&存储条件

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