BAN ORL 24 |CAS:1401463-54-4 Probechem Biochemicals

Chemical Structure : BAN ORL 24

CAS No.: 1401463-54-4

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BAN ORL 24 (BAN-ORL-24;BAN ORL-24)

货号: PC-43402Not For Human Use, Lab Use Only.

BAN ORL 24 is a potent, selective, non-peptide nociceptin/orphanin FQ receptor (NOP receptor, ORL1) antagonist with IC50 of 0.27 nM, displays no significant activity for κ-, μ- and δ-receptors.

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10 mg	￥1180	In stock
25 mg	￥1980	In stock
50 mg	￥3280	In stock
100 mg		Get quote

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生物&药学活性

BAN ORL 24 is a potent, selective, non-peptide nociceptin/orphanin FQ receptor (NOP receptor, ORL1) antagonist with IC50 of 0.27 nM, displays no significant activity for κ-, μ- and δ-receptors.
BAN ORL 24 produces a concentration-dependent displacement of [(3)H]N/OFQ binding to CHO(hNOP) cell membranes with pKi of 9.62 and selectivity (1000 fold) over classical opioid receptors.
BAN ORL 24 antagonizes the pronociceptive and antinociceptive effects of N/OFQ in vivo.

物理化学性质&存储条件

分子量	506.5076
分子式	C27H37Cl2N3O2
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	2-Pyrrolidinecarboxamide, 1-(phenylmethyl)-N-(3-spiro[isobenzofuran-1(3H),4'-piperidin]-1'-ylpropyl)-, (2R)-

参考文献

1. Fischetti C, et al. Eur J Pharmacol. 2009 Jul 1;614(1-3):50-7.

BAN ORL 24 (BAN-ORL-24;BAN ORL-24)

生物&药学活性

物理化学性质&存储条件

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BAN ORL 24 (BAN-ORL-24;BAN ORL-24)

生物&药学活性

物理化学性质&存储条件

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