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首页-小分子抑制剂&激动剂-GPCR-5-HT Receptor-Astemizole
Astemizole

Chemical Structure : Astemizole

CAS No.: 68844-77-9

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Astemizole (R43512, R 43512)

货号: PC-28213Not For Human Use, Lab Use Only.

Astemizole (R43512) is a second-generation histamine H1-receptor antagonist with IC50 of 4 nM, also shows potent hERG K+ channel blocking activity with IC50 of 0.9 nM.

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50 mg ￥880 In stock
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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

Astemizole (R43512) is a second-generation histamine H1-receptor antagonist with IC50 of 4 nM, also shows potent hERG K+ channel blocking activity with IC50 of 0.9 nM.

物理化学性质&存储条件

分子量 458.58
分子式 C28H31FN4O
外观性状 Solid
CAS No.
储存条件
固体粉末
-20°C 12 个月; 4°C 6 个月
配置液
-80°C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

1-(4-Fluorobenzyl)-N-(1-(4-methoxyphenethyl)piperidin-4-yl)-1H-benzo[d]imidazol-2-amine

参考文献

1. Nicholson AN, et al. Br J Clin Pharmacol. 1982 Nov;14(5):683-90.

2. Laduron PM, et al. Mol Pharmacol. 1982 Mar;21(2):294-300.

3. Suessbrich H, et al. FEBS Lett. 1996 Apr 29;385(1-2):77-80.

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