Alvimopan | μ-opioid receptor antagonist | Probechem Biochemicals

Chemical Structure : Alvimopan

CAS No.: 156053-89-3

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Alvimopan (ADL 8-2698, LY246736)

货号: PC-43423Not For Human Use, Lab Use Only.

Alvimopan (LY 246736) is a selective peripherally acting μ-opioid (MOR) antagonist with IC50 of 1.7 nM for the treatment of postoperative ileus.

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生物&药学活性

Alvimopan (LY 246736) is a selective peripherally acting μ-opioid (MOR) antagonist with IC50 of 1.7 nM for the treatment of postoperative ileus.
Alvimopan (LY 246736) prevents gastrointestinal effects of intravenous morphine without affecting analgesia.
Alvimopan (LY 246736) is orally active.

物理化学性质&存储条件

分子量	424.5326
分子式	C25H32N2O4
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	Glycine, N-[(2S)-2-[[(3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethyl-1-piperidinyl]methyl]-1-oxo-3-phenylpropyl]-

参考文献

1. Fukuda H, et al. Brain Res. 2006 Aug 2;1102(1):63-70.

2. Taguchi A, et al. N Engl J Med. 2001 Sep 27;345(13):935-40.

3. Schmidt WK. Am J Surg. 2001 Nov;182(5A Suppl):27S-38S.

Alvimopan (ADL 8-2698, LY246736)

生物&药学活性

物理化学性质&存储条件

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Alvimopan (ADL 8-2698, LY246736)

生物&药学活性

物理化学性质&存储条件

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