Aliskiren |CAS:173334-57-1 Probechem Biochemicals

Chemical Structure : Aliskiren

CAS No.: 173334-57-1

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Aliskiren (CGP 60536;CGP60536B;SPP 100)

货号: PC-42905Not For Human Use, Lab Use Only.

Aliskiren (CGP60536B) is a first-in-class, potent and highly selective, direct renin inhibitor with IC50 of 0.6 nM.

规格	价格	库存
5 mg	￥680	In stock
10 mg	￥980	In stock
25 mg	￥1580	In stock
50 mg	￥2480	In stock
100 mg		Get quote

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生物&药学活性

Aliskiren (CGP60536B) is a first-in-class, potent and highly selective, direct renin inhibitor with IC50 of 0.6 nM.
Aliskiren shows no significant inhibition on Cathepsin D, Cathepsin E, Pepsin and HIV-1 peptidase (> 50 uM); orally bioactive.

物理化学性质&存储条件

分子量	551.7583
分子式	C30H53N3O6
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	Benzeneoctanamide, .delta.-amino-N-(3-amino-2,2-dimethyl-3-oxopropyl)-.gamma.-hydroxy-4-methoxy-3-(3-methoxypropoxy)-.alpha.,.zeta.-bis(1-methylethyl)-, (.alpha.S,.gamma.S,.delta.S,.zeta.S)-

参考文献

1. Wood JM, et al. Biochem Biophys Res Commun. 2003 Sep 5;308(4):698-705.

2. Desjarlais M, et al. Atherosclerosis. 2015 Oct;242(2):450-60.

3. Jumar A, et al. J Hypertens. 2015 Dec;33(12):2491-9.

Aliskiren (CGP 60536;CGP60536B;SPP 100)

生物&药学活性

物理化学性质&存储条件

参考文献

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Aliskiren (CGP 60536;CGP60536B;SPP 100)

生物&药学活性

物理化学性质&存储条件

参考文献

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