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首页-小分子抑制剂&激动剂-Metabolic Enzyme/Protease-11β-HSD-AZD 8329
AZD 8329

Chemical Structure : AZD 8329

CAS No.: 1048668-70-7

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AZD 8329 (AZD8329)

货号: PC-62766Not For Human Use, Lab Use Only.

AZD8329 is a potent, selective 11β-HSD1 inhibitor with IC50 of 9 nM, displays excellent selectivity versus relatedd 11β-HSD2, 17β-HSD1 and 17β-HSD3 (IC50>30 uM).

规格 价格 库存 数量
5 mg ￥1980 In stock
10 mg ￥2980 In stock
25 mg ￥4980 In stock
50 mg Get quote
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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

AZD8329 is a potent, selective 11β-HSD1 inhibitor with IC50 of 9 nM, displays excellent selectivity versus relatedd 11β-HSD2, 17β-HSD1 and 17β-HSD3 (IC50>30 uM).
AZD8329 shows significantly reduced acyl glucuronidation liability compared with AZD4017.

物理化学性质&存储条件

分子量 421.541
分子式 C25H31N3O3
外观性状 Solid
CAS No.
储存条件
固体粉末
-20 °C 12 个月; 4°C 6 个月
配置液
-80 °C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

4-[4-(2-adamantylcarbamoyl)-5-tert-butyl-pyrazol-1-yl]benzoic acid

参考文献

1. Scott JS, et al. J Med Chem. 2012 Nov 26;55(22):10136-47.

2. Morentin Gutierrez P, et al. Br J Pharmacol. 2015 Oct;172(20):4806-16.

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