ARUK2001607 | PI5P4Kγ inhibitor | Probechem Biochemicals

Chemical Structure : ARUK2001607

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ARUK2001607 (ARUK 2001607)

货号: PC-49589Not For Human Use, Lab Use Only.

ARUK2001607 is a potent, selective and brain penetrant PI5P4Kγ inhibitor with binding KD of 7.1 nM, pIC50 of 7.1 (PI5P4Kγ+).

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生物&药学活性

ARUK2001607 is a potent, selective and brain penetrant PI5P4Kγ inhibitor with binding KD of 7.1 nM, pIC50 of 7.1 (PI5P4Kγ+).
ARUK2001607 showed excellent selectivity data against >150 kinases and a Cerep safety panel, also showed good potencies at PI5P4Kγ (WT and γ+), were selective vs PI5P4Kα and β.

物理化学性质&存储条件

分子量	319.40
分子式	C14H13N3O2S2
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	6-Methyl-N-(4-(methylsulfonyl)phenyl)thieno[2,3-d]pyrimidin-4-amine

参考文献

1. Timothy P C Rooney, et al. J Med Chem. 2022 Dec 14. doi: 10.1021/acs.jmedchem.2c01693.

ARUK2001607 (ARUK 2001607)

生物&药学活性

物理化学性质&存储条件

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ARUK2001607 (ARUK 2001607)

生物&药学活性

物理化学性质&存储条件

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