APJ agonist 47

Chemical Structure : APJ agonist 47

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货号: PC-38748Not For Human Use, Lab Use Only.

APJ agonist 47 is a potent and selective, orally active apelin receptor (APJ) agonist EC50 of 6.5 nM.

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生物&药学活性

APJ agonist 47 is a potent and selective, orally active apelin receptor (APJ) agonist EC50 of 6.5 nM.
APJ agonist 47 has vastly reduced brain penetration and is devoid of significant off-target liability.
APJ agonist 47 is suitable for in vivo studies of APJ in peripheral tissues after oral administration.

物理化学性质&存储条件

分子量	566.581
分子式	C26H31F5N8O
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(S)-1-cyclopentyl-N-(4-(3,3-difluoropiperidin-1-yl)-1-(1H-tetrazol-5-yl)butan-2-yl)-5-(2-(trifluoromethyl)phenyl)-1H-pyrazole-3-carboxamide

参考文献

1. Sanju Narayanan, et al. Bioorg Med Chem. 2022 May 6;66:116789.

APJ agonist 47

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物理化学性质&存储条件

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APJ agonist 47

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物理化学性质&存储条件

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