AM-5262 |CAS:1222088-90-5 Probechem Biochemicals

首页-小分子抑制剂&激动剂-GPCR-Free Fatty Acid Receptor (FFAR)-AM-5262

Chemical Structure : AM-5262

加入收藏

AM-5262 (AM5262)

货号: PC-63042Not For Human Use, Lab Use Only.

AM-5262 is a potent full GPR40 (FFA1) agonist with EC50 of 81 nM.

规格	价格	库存	数量
25 mg		Get quote
50 mg		Get quote
100 mg		Get quote
250 mg		Get quote

获取报价单

* 请选择数量再加入购物车

or Bulk Inquiry

大包装，大折扣！

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

AM-5262 is a potent full GPR40 (FFA1) agonist with EC50 of 81 nM.
AM-5262 shows improved rat PK profile and general selectivity profile, enhances glucose stimulated insulin secretion (mouse and human islets) and improves glucose homeostasis in vivo (OGTT in HF/STZ mice) when compared to AM-1638.

物理化学性质&存储条件

分子量	514.637
分子式	C33H35FO4
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(1R,2R)-6'-((2-((R)-2,2-dimethylcyclopentyl)-2'-fluoro-5'-methoxy-[1,1'-biphenyl]-4-yl)methoxy)-2',3'-dihydrospiro[cyclopropane-1,1'-indene]-2-carboxylic acid

参考文献

1. Wang Y, et al. ACS Med Chem Lett. 2013 May 7;4(6):551-5.

联系我们 sales@probechem.com

AM-5262 (AM5262)

生物&药学活性

物理化学性质&存储条件

参考文献

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

询单

AM-5262 (AM5262)

生物&药学活性

物理化学性质&存储条件

参考文献

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

询单

Get Quotation Now

* Indicates a Required FieldYour information is safe with us.