AH6809 | PGD2 antagonist | Probechem Biochemicals

Chemical Structure : AH6809

CAS No.: 33458-93-4

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AH6809 (AH-6809)

货号: PC-42574Not For Human Use, Lab Use Only.

AH6809 is a xanthone derivative that fuctions as an EP and DP receptor antagonist with Ki of 1217, 1150, 1597, and 1415 nM for the cloned human EP1, EP2, EP3-III, and DP receptor respectively.

规格	价格	库存
10 mg	￥1280	In stock
25 mg	￥2180	In stock
50 mg	￥3580	In stock
100 mg	￥5280	In stock
250 mg		Get quote

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生物&药学活性

AH6809 is a xanthone derivative that fuctions as an EP and DP receptor antagonist with Ki of 1217, 1150, 1597, and 1415 nM for the cloned human EP1, EP2, EP3-III, and DP receptor respectively.
AH6809 blocks the PGE2-induced accumulation of cAMP in COS cells transfected with the human EP2 receptor。
AH6809 is an effective antagonist antiaggregatory actions of PGD2, but not PGI2, with EC50 50 uM in whole human platelet.

物理化学性质&存储条件

分子量	298.2901
分子式	C17H14O5
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	9H-Xanthene-2-carboxylic acid, 6-(1-methylethoxy)-9-oxo-

参考文献

1. Armstrong RA, et al. Br J Pharmacol. 1986 Mar;87(3):543-51.

2. Woodward DF, et al. Biochem Pharmacol. 1995 Nov 9;50(10):1731-3.

3. Keery RJ, et al. Br J Pharmacol. 1988 Jul;94(3):745-54.

AH6809 (AH-6809)

生物&药学活性

物理化学性质&存储条件

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AH6809 (AH-6809)

生物&药学活性

物理化学性质&存储条件

参考文献

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